Clinical Investigation of Tyrosinase Inhibitors: Past, Present, and Future [0.03%]
酪氨酸酶抑制剂的临床研究：过去、现在和未来展望
Yuanyuan Wang,Ruijia Jiang,Baichen Xiong et al.
Yuanyuan Wang et al.
Tyrosinase (EC 1.14.18.1) is a pivotal enzyme that catalyzes the conversion of L-tyrosine to dopaquinone through a dual oxidation process, initiating melanin biosynthesis. Melanin plays a critical role in various biological processes, and i...
Natural Mimetic 4,6-dihydroxyaurone Derivatives as Tyrosinase Inhibitors: Design, Synthesis, and Biological Evaluation [0.03%]
天然拟效的4,6-羟基黄酮衍生物作为酪氨酸酶抑制剂：设计，合成及生物活性评价
Quoc-Thai Nguyen,Giao Quynh Tran,Huy Thanh Ta et al.
Quoc-Thai Nguyen et al.
Introduction: Tyrosinase, a key enzyme in melanin biosynthesis and food browning, has become an important target for inhibitor development. Aim: ...
Tyrosinase Inhibitors Among Flora of Lubelskie Region-Application of Bio-Chromatographic Approach and Zebrafish Model in Bioactivity Screening of Plant Material [0.03%]
利用生物色谱法和斑马鱼模型筛选植物样品的活性以发现卢贝林省植物资源中的酪氨酸酶抑制剂
Kamila Kusio-Targońska,Nataliia Kosheva,Krzysztof Kamil Wojtanowski et al.
Kamila Kusio-Targońska et al.
The whitening potential of natural products is commonly assessed through spectrophotometric assays that colorimetrically measure the inhibitory effects on tyrosinase, a key enzyme in pigment formation. However, these assays fail to provide ...
One-pot four-component synthesis of some novel hydrazone-Schiff bases of polyhydroquinoline as potent tyrosinase inhibitors: in vitro, molecular docking and simulations approaches [0.03%]
一种新的单锅四组分合成多氢喹啉衍生物 Hydrazone-Schiff 醌的研究：体外实验，分子对接和理论计算方法学研究
Sajjad Ur Rahman,Muhammad Naveed Umar,Aftab Alam et al.
Sajjad Ur Rahman et al.
Seventeen novel polyhydroquinoline (1) based Schiff bases (4-20) were synthesized in excellent yields through Hantzsch reaction, characterized by means of spectroscopic techniques and finally screened for their in vitro tyrosinase inhibitor...
Design, synthesis and biological evaluation of novel kojic acid triazole hybrids as tyrosinase inhibitors and antibrowning agents [0.03%]
新型曲酸三唑衍生物的合成及对酪氨酸酶抑制和抗褐变作用的研究
Dan Liu,Junyuan Tang,Sheng Tao et al.
Dan Liu et al.
In this study, two series of kojic acid triazole hybrids, namely 6a-6p and 13a-13t, were designed and synthesized. Subsequently, their biological activities including anti-tyrosinase, antioxidant, and as anti-browning effects were investiga...
New Record of Potential Tyrosinase Inhibitory, Antioxidant and Photoprotective Effects of Vietnamese Castanea mollissima Extracts [0.03%]
越南栗子提取物新的多酚记录及其潜在的酪氨酸酶抑制、抗氧化和光防护作用
Thi Thu Le Vu,San-Lang Wang,Tan Luc Quang et al.
Thi Thu Le Vu et al.
In this study, the potential anti-tyrosinase, antioxidant, and UV absorption efficiency of the extracts of different parts of Castanea mollissima were evaluated. The leaf extract exhibited the most potential antioxidant effect with DPPH and...
Unveiling tyrosinase inhibition: exploring secondary metabolites from Fernandoa adenophylla through biological screening and molecular docking [0.03%]
基于生物筛选和分子对接技术从 Fernandoa adenophylla 中探索次要代谢物及其酪氨酸酶抑制作用研究
Abdur Rauf,Umer Rashid,Zuneera Akram et al.
Abdur Rauf et al.
The current study investigated the tyrosinase inhibitory activity of compounds extracted from Fernandoa adenophylla, complemented by in silico analysis. Using methanolic extract and chromatography, several compounds were isolated and tested...
Isoindole-1,3-Dione Sulfonamides as Potent Inhibitors of Glucosidase, Aldose Reductase, and Tyrosinase: A Molecular Docking and Enzyme Inhibition Study [0.03%]
异吲哚-1,3-二酮磺酰胺类葡萄糖苷酶、醛还原酶和酪氨酸酶的高效抑制剂：分子对接及酶抑制研究
Zozan Aslan,Esra Yılmaz,Nurgül Pulat et al.
Zozan Aslan et al.
Diabetes mellitus, especially type 2, is a global health challenge, and effective enzyme inhibitors are essential for its control. Conventional inhibitors have drawbacks such as gastrointestinal side effects and regional availability, examp...
Innovative dopamine-modified carbon quantum dot fluorescence sensor meets affinity chromatography: A breakthrough in Tyrosinase inhibitor screening in food [0.03%]
创新型多巴胺改性碳量子点荧光传感器结合亲和层析在食品酪氨酸酶抑制剂筛查中的突破
Tao Gao,Weibiao Wang,Mei Wang et al.
Tao Gao et al.
Tyrosinase (TYR), a polyphenol oxidase crucial for melanin synthesis, plays various biological functions, and its inhibitors are widely used in the cosmetics and food industries for skin-lightening and anti-browning applications. Here, an i...
Efficacy of Natural Products as Tyrosinase Inhibitors in Hyperpigmentation Therapy: Anti-Melanogenic or Antibrowning Effects [0.03%]
天然产物作为酪氨酸酶抑制剂在色素沉着治疗中的功效：抗黑素生成或抗棕化作用
Mahrous H Mahrous,Shymaa Abdel-Dayem,Islam M Adel et al.
Mahrous H Mahrous et al.
Hyperpigmentation in human skin and enzymatic browning are prevalent and undesirable phenomena. Tyrosinase, the principal enzyme implicated in these processes, is recognized for its crucial role in melanogenesis and browning reactions. This...
耗时 0.22046 秒，为您在
48229835
条记录里面共找到 686 篇文章 [XML]