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Tetracyclic triterpenes from Chios Mastic Gum act as TGR5 and RORγ modulators

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Background: Chios mastic gum (CMG) is a natural resin from Pistacia lentiscus L. var. Chia (Anacardiaceae). It contains high concentrations of triterpenoids, with 24Z-masticadienonic acid (24Z-MNA) and 24Z-isomasticadienonic acid... ...