Degraders of histone lysine methyltransferases: Progress, challenges, and opportunities
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Histone lysine methyltransferases (HKMTs) are a class of enzymes capable of catalyzing the methylation modification of lysine residues on histones. Members of the lysine methyltransferase family, such as EZH2, G9a, DOT1L, NSD2, NSD3, and ASH1L, show overexpres... ...
