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Recent patent landscape of ASK1 inhibitors: spotlight on 2-(1-isopropyl-4H-1,2,4-triazole-3-yl) pyridine as a privileged scaffold

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Introduction: Apoptosis signal-regulating kinase 1 (ASK1) is an important stress-responsive kinase involved in multiple pathological conditions including fibrosis, cancer, cardiovascular disorders, inflammatory diseases, and neur... ...