Antiallodynic effect of a novel sigma-1 receptor antagonist N-(1-benzylpiperidin-4-yl)-2,4-dichlorobenzamide (Dicloperidine): Synthesis and combined bioevaluation
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This study describes the synthesis and combined biological evaluation (in silico, in vitro, and in vivo) of N-(1-benzylpiperidin-4-yl)-2,4-dichlorobenzamide (Dicloperidine), a novel analogue structurally related to compound LMH-2 and haloperidol, both stablish... ...