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Optimizing [99mTc]Tc-Tamsulosin for Enhanced Tumor Detection: A Comprehensive Approach from Preparation to In Vivo Evaluation

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Purpose: To investigate the potential of Tamsulosin hydrochloride, a selective α1-adrenoceptor antagonist, as a tumor-targeting ligand when labeled with Technetium-99 m [⁹⁹ᵐTc] for use as a novel radiopharmaceutical. This stu... ...