A simple solid-phase approach for the synthesis of DOTA-conjugated α-ketoamide-based fibroblast activation protein-targeted ligands
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Several studies have shown that fibroblast activation protein (FAP)-targeted radioligands with an α-ketoamide as the warhead can lead to high affinity for FAP and prolonged tumor retention. However, the preparation of reported FAP-targeted ligands requires mu... ...
