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Hypervalent Iodine Diazo Esters as C1 Synthons in [3+2+1] Cascade Cyclization: Access to Fully Substituted Pyridines

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Fully substituted pyridines are important cores in natural products, functional materials, and pharmaceuticals. Building such a motif usually requires multiple steps, a transition metal as a catalyst, and external additives. Herein, a [3+2+1] cascade annulatio... ...