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Zoomlab™-Guided Co-crystal Engineering of Nilotinib for Improved Dissolution

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Nilotinib (NH), a second-generation tyrosine kinase inhibitor for chronic myelogenous leukemia (CML), exhibits poor aqueous solubility and low intestinal permeability, classifying it as a Biopharmaceutics Classification System (BCS) Class IV drug. This study a... ...