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Androgen receptor blockade and its effect on PSMA-localization in prostate cancer: Implications for radioligand therapy

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Prostate-specific membrane antigen (PSMA) is a key target for radioligand therapy (RLT) in prostate cancer (PCa). However, its subcellular localization is critical, as ligand uptake via PSMA mediated endocytosis influences therapeutic efficacy. This study exam... ...