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Induction of P-glycoprotein overexpression in brain endothelial cells as a model to study blood-brain barrier efflux transport

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The blood-brain barrier (BBB) is comprised of specialized brain endothelial cells (BECs) that contribute to maintaining central nervous system (CNS) homeostasis. BECs possess properties such as an array of multi-drug efflux transporters that eject various drug... ...