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Emerging TSPO-PET Radiotracers for Imaging Neuroinflammation: A Critical Analysis

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The translocator protein (TSPO) is a biomarker for imaging neuroinflammation via Positron Emission Tomography (PET) across a broad range of CNS conditions. Most clinically used PET ligands targeting TSPO have limitations, including high lipophilicity and off-t... ...