Rational Search for Betaine/GABA Transporter 1 Inhibitors─ In Vitro Evaluation of Selected Hit Compound
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Inhibitory neurotransmission mediated by γ-aminobutyric acid (GABA) plays an important role in maintaining body homeostasis. Disturbances in GABA signaling are implicated in a multitude of neurologic and psychiatric conditions, including epilepsy, ischemia, a... ...