Conformationally constrained analogs of BAY 59-3074 as novel cannabinoid receptor ligands
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To obtain information on the pharmacophoric requirements of the CB1/CB2 partial agonist BAY 59-3074 we have synthesized a series of new conformationally constrained dibenzofuran (4a-d) and dibenzopyran analogs (5). All constrained analogs exhibited reduced bin... ...
